PDB Entry - 10HY (pdb_000010hy)

(Status - Released)

Summary information:

Title: Structure of CHK1 10-pt. mutant complex with macrocyclic LRRK2 inhibitor compound 1 ((11R)-8-chloro-3,11-dimethyl-2-(oxan-4-yl)-2,4,10,11,12,13-hexahydro-9,5-(azeno)pyrazolo[3,4-b][1,4,6,10]oxatriazacyclotridecine)

PDB DOI: https://doi.org/10.2210/pdb10hy/pdb

Primary publication DOI: https://doi.org/10.1021/acs.jmedchem.6c00238

Entry authors: Palte, R.L., Yu, E.C., Zhou, H.

Initial deposition on: 21 January 2026

Initial release on: 8 April 2026

Latest revision on: 8 April 2026

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Structure coordinates (PDBx/mmCIF)

Structure coordinates (PDBML)

X-ray diffraction data (PDBx/mmCIF)

Validation report (PDF)

Validation report (mmCIF)

Validation report (XML)

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