PDB Entry - 10JT (pdb_000010jt)

(Status - Released)

Summary information:

Title: CRYSTAL STRUCTURE OF KIRSTEN RAT SARCOMA G12C COMPLEXED WITH GMPPNP AND COVALENTLY BOUND TO 1-[(2R,3R)-3-{[(7P)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoro-2-{ [(2R,4R,7aS)-2-fluorotetrahydro-1H-pyrrolizin-7a(5H)-yl]methoxy}pyrido[4,3-d] pyrimidin-4-yl](methyl)amino}-2-methylpyrrolidin-1-yl]-3-(pyrazin-2-yl)propan-1-one

PDB DOI: https://doi.org/10.2210/pdb10jt/pdb

Entry authors: Sheriff, S.

Initial deposition on: 22 January 2026

Initial release on: 4 March 2026

Latest revision on: 4 March 2026

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Structure coordinates (PDBx/mmCIF)

Structure coordinates (PDBML)

X-ray diffraction data (PDBx/mmCIF)

Validation report (PDF)

Validation report (mmCIF)

Validation report (XML)

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