PDB Entry - 1EAS (pdb_00001eas)

(Status - Released)

Summary information:

Title: NONPEPTIDIC INHIBITORS OF HUMAN LEUKOCYTE ELASTASE. 3. DESIGN, SYNTHESIS, X-RAY CRYSTALLOGRAPHIC ANALYSIS, AND STRUCTURE-ACTIVITY RELATIONSHIPS FOR A SERIES OF ORALLY ACTIVE 3-AMINO-6-PHENYLPYRIDIN-2-ONE TRIFLUOROMETHYL KETONES

PDB DOI: https://doi.org/10.2210/pdb1eas/pdb

Primary publication DOI: https://doi.org/10.1021/jm00046a016

Entry authors: Ceccarelli, C.

Initial deposition on: 22 November 1994

Initial release on: 7 February 1995

Latest revision on: 9 October 2024

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Structure coordinates (PDBx/mmCIF)

Structure coordinates (PDB)

Structure coordinates (PDBML)

X-ray diffraction data (PDBx/mmCIF)

Validation report (PDF)

Validation report (XML)

Validation report (mmCIF)

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