PDB Entry - 1PYN

(Status - Released)

Summary information:

Title: DUAL-SITE POTENT, SELECTIVE PROTEIN TYROSINE PHOSPHATASE 1B INHIBITOR USING A LINKED FRAGMENT STRATEGY AND A MALONATE HEAD ON THE FIRST SITE

PDB DOI: https://doi.org/10.2210/pdb1pyn/pdb

Primary publication DOI: https://doi.org/10.1016/S0960-894X(03)00725-X

Entry authors: Szczepankiewicz, B.G., Liu, G., Hajduk, P.J., Abad-Zapatero, C., Zhonghua, P., Lubben, T., Trevillyan, J.M., Stashko, M., Ballaron, S.J., Liang, H.

Initial deposition on: 9 July 2003

Initial release on: 16 September 2003

Latest revision on: 16 August 2023

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