PDB Entry - 3RKZ

(Status - Released)

Summary information:

Title: Discovery of a stable macrocyclic o-aminobenzamide Hsp90 inhibitor capable of significantly decreasing tumor volume in a mouse xenograft model.

PDB DOI: https://doi.org/10.2210/pdb3rkz/pdb

Primary publication DOI: https://doi.org/10.1016/j.bmcl.2011.05.102

Entry authors: Zapf, C.W., Bloom, J.D., Li, Z., Dushin, R.G., Nittoli, T., Otteng, M., Nikitenko, A., Golas, J.M., Liu, H., Lucas, J., Boschelli, F., Vogan, E., Olland, A., Johnson, M., Levin, J.I.

Initial deposition on: 18 April 2011

Initial release on: 13 July 2011

Latest revision on: 13 September 2023

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Structure coordinates (PDB)

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