PDB Entry - 3K5K

(Status - Released)

Summary information:

Title: Discovery of a 2,4-Diamino-7-aminoalkoxy-quinazoline as a Potent Inhibitor of Histone Lysine Methyltransferase, G9a

PDB DOI: https://doi.org/10.2210/pdb3k5k/pdb

Primary publication DOI: https://doi.org/10.1021/jm901543m

Entry authors: Dong, A., Wasney, G.A., Liu, F., Chen, X., Allali-Hassani, A., Senisterra, G., Chau, I., Bountra, C., Weigelt, J., Edwards, A.M., Arrowsmith, C.H., Frye, S.V., Bochkarev, A., Brown, P.J., Jin, J., Vedadi, M., Structural Genomics Consortium (SGC)

Initial deposition on: 7 October 2009

Initial release on: 10 November 2009

Latest revision on: 6 September 2023

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Structure coordinates (PDBML)

Structure coordinates (PDB)

X-ray diffraction data (PDBx/mmCIF)

Validation report (PDF)

Validation report (XML)

Validation report (mmCIF)

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