PDB Entry - 3R92

(Status - Released)

Summary information:

Title: Discovery of a macrocyclic o-aminobenzamide Hsp90 inhibitor with heterocyclic tether that shows extended biomarker activity and in vivo efficacy in a mouse xenograft model.

PDB DOI: https://doi.org/10.2210/pdb3r92/pdb

Primary publication DOI: https://doi.org/10.1016/j.bmcl.2011.04.102

Entry authors: Zapf, C.W., Bloom, J.D., McBean, J.L., Dushin, R.G., Golas, J.M., Liu, H., Lucas, J., Boschelli, F., Vogan, E.M., Levin, J.I.

Initial deposition on: 24 March 2011

Initial release on: 8 June 2011

Latest revision on: 21 February 2024

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Structure coordinates (PDB)

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