PDB Entry - 3VAP

(Status - Released)

Summary information:

Title: Synthesis and SAR Studies of imidazo-[1,2-a]-pyrazine Aurora kinase inhibitors with improved off target kinase selectivity

PDB DOI: https://doi.org/10.2210/pdb3vap/pdb

Primary publication DOI: https://doi.org/10.1016/j.bmcl.2012.03.051

Entry authors: Voss, M.E., Rainka, M.P., Fleming, M., Peterson, L.H., Belanger, D.B., Siddiqui, M.A., Hruza, A., Voigt, J., Basso, A.D., Gray, K.

Initial deposition on: 29 December 2011

Initial release on: 2 May 2012

Latest revision on: 28 February 2024

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