PDB Entry - 3WZJ

(Status - Released)

Summary information:

Title: CRYSTAL STRUCTURE OF HUMAN MPS1 CATALYTIC DOMAIN IN COMPLEX WITH 4-(6-(cyclohexylamino)-8-(((tetrahydro-2H-pyran-4-yl)methyl)amino)imidazo[1,2-b]pyridazin-3-yl)-N-cyclopropylbenzamide

PDB DOI: https://doi.org/10.2210/pdb3wzj/pdb

Primary publication DOI: https://doi.org/10.1021/jm501599u

Entry authors: Kusakabe, K., Ide, N., Daigo, Y., Itoh, T., Yamamoto, T., Kojima, E., Mitsuoka, Y., Tadano, G., Tagashira, S., Higashino, K., Okano, Y., Sato, Y., Inoue, M., Iguchi, M., Kanazawa, T., Ishioka, Y., Dohi, K., Kido, Y., Sakamoto, S., Ando, S., Maeda, M., Higaki, M., Yoshizawa, H., Mura, H., Nakamura, Y.

Initial deposition on: 29 September 2014

Initial release on: 11 February 2015

Latest revision on: 24 August 2022

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