PDB Entry - 4ISE

(Status - Released)

Summary information:

Title: Human glucokinase in complex with novel activator (2S)-3-cyclohexyl-2-(6-fluoro-4-oxoquinazolin-3(4H)-yl)-N-(1,3-thiazol-2-yl)propanamide

PDB DOI: https://doi.org/10.2210/pdb4ise/pdb

Primary publication DOI: https://doi.org/10.1016/j.bmcl.2013.01.093

Entry authors: Hosfield, D., Skene, R.J.

Initial deposition on: 16 January 2013

Initial release on: 20 March 2013

Latest revision on: 28 February 2024

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Structure coordinates (PDBML)

Structure coordinates (PDB)

X-ray diffraction data (PDBx/mmCIF)

Validation report (mmCIF)

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Validation report (PDF)

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