PDB Entry - 4K8S (pdb_00004k8s)

(Status - Released)

Summary information:

Title: Hydroxyethylamine-based inhibitors of BACE1: P1-P3 macrocyclization can improve potency, selectivity, and cell activity

PDB DOI: https://doi.org/10.2210/pdb4k8s/pdb

Primary publication DOI: https://doi.org/10.1016/j.bmcl.2013.05.028

Entry authors: Jordan, S.R.

Initial deposition on: 18 April 2013

Initial release on: 10 July 2013

Latest revision on: 16 October 2024

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Structure coordinates (PDB)

Structure coordinates (PDBML)

X-ray diffraction data (PDBx/mmCIF)

Validation report (mmCIF)

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