PDB Entry - 4C66

(Status - Released)

Summary information:

Title: Discovery of Epigenetic Regulator I-BET762: Lead Optimization to Afford a Clinical Candidate Inhibitor of the BET Bromodomains

PDB DOI: https://doi.org/10.2210/pdb4c66/pdb

Primary publication DOI: https://doi.org/10.1021/JM401088K

Entry authors: Chung, C., Mirguet, O.

Initial deposition on: 17 September 2013

Initial release on: 2 October 2013

Latest revision on: 30 October 2013

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Structure coordinates (PDBx/mmCIF)

Structure coordinates (PDBML)

Structure coordinates (PDB)

X-ray diffraction data (PDBx/mmCIF)

Validation report (PDF)

Validation report (XML)

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