PDB Entry - 4ER3
(Status - Released)Summary information:
Title: Crystal Structure of Human DOT1L in complex with inhibitor EPZ004777
PDB DOI: https://doi.org/10.2210/pdb4er3/pdb
Primary publication DOI: https://doi.org/10.1038/ncomms2304
Entry authors: Wernimont, A.K., Tempel, W., Yu, W., Scopton, A., Li, Y., Nguyen, K.T., Federation, A., Marineau, J., Qi, J., Vedadi, M., Bradner, J.E., Schapira, M., Arrowsmith, C.H., Edwards, A.M., Bountra, C., Brown, P.J., Structural Genomics Consortium (SGC)
Initial deposition on: 19 April 2012
Initial release on: 16 May 2012
Latest revision on: 28 February 2024
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Structure coordinates (PDBx/mmCIF)
Structure coordinates (PDBML)
Structure coordinates (PDB)
X-ray diffraction data (PDBx/mmCIF)
Validation report (mmCIF)
Validation report (PDF)
Validation report (XML)
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