PDB Entry - 4F09

(Status - Released)

Summary information:

Title: Discovery and Optimization of C-2 Methyl Imidazo-pyrrolopyridines as Potent and Orally Bioavailable JAK1 Inhibitors with Selectivity over JAK2

PDB DOI: https://doi.org/10.2210/pdb4f09/pdb

Primary publication DOI: https://doi.org/10.1021/jm300628c

Entry authors: Murray, J.M.

Initial deposition on: 3 May 2012

Initial release on: 4 July 2012

Latest revision on: 6 December 2023

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Structure coordinates (PDBx/mmCIF)

Structure coordinates (PDBML)

Structure coordinates (PDB)

X-ray diffraction data (PDBx/mmCIF)

Validation report (XML)

Validation report (PDF)

Validation report (mmCIF)

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