PDB Entry - 4GPJ

(Status - Released)

Summary information:

Title: Crystal Structure of the first bromodomain of human BRD4 in complex with a isoxazolylbenzimidazole ligand

PDB DOI: https://doi.org/10.2210/pdb4gpj/pdb

Primary publication DOI: https://doi.org/10.1039/C2MD20189E

Entry authors: Filippakopoulos, P., Picaud, S., Qi, J., Felletar, I., Heightman, T.D., Brennan, P., von Delft, F., Bountra, C., Arrowsmith, C.H., Edwards, A., Knapp, S., Structural Genomics Consortium (SGC)

Initial deposition on: 21 August 2012

Initial release on: 17 October 2012

Latest revision on: 13 September 2023

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Structure coordinates (PDBx/mmCIF)

Structure coordinates (PDBML)

Structure coordinates (PDB)

X-ray diffraction data (PDBx/mmCIF)

Validation report (mmCIF)

Validation report (XML)

Validation report (PDF)

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