PDB Entry - 4JNM

(Status - Released)

Summary information:

Title: Discovery of Potent and Efficacious Urea-containing Nicotinamide Phosphoribosyltransferase (NAMPT) Inhibitors with Reduced CYP2C9 Inhibition Properties

PDB DOI: https://doi.org/10.2210/pdb4jnm/pdb

Primary publication DOI: https://doi.org/10.1016/j.bmcl.2013.04.040

Entry authors: Gunzner-Toste, J., Zhao, G., Bauer, P., Baumeister, T., Buckmelter, A.J., Caligiuri, M., Clodfelter, K.H., Fu, B., Han, B., Ho, Y., Kley, N., Liederer, B., Lin, J., Mukadam, S., O'Brien, T., Reynolds, D.J., Sharma, G., Skelton, N., Smith, C.C., Oh, A., Wang, W., Wang, Z., Xiao, Y., Yuen, P., Zak, M., Zhang, L., Zheng, X., Bair, K.W., Dragovich, P.S.

Initial deposition on: 15 March 2013

Initial release on: 29 May 2013

Latest revision on: 28 February 2024

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