PDB Entry - 4LV9

(Status - Released)

Summary information:

Title: Fragment-based Identification of Amides Derived From trans-2-(Pyridin-3-yl)cyclopropanecarboxylic Acid as Potent Inhibitors of Human Nicotinamide Phosphoribosyltransferase (NAMPT)

PDB DOI: https://doi.org/10.2210/pdb4lv9/pdb

Primary publication DOI: https://doi.org/10.1016/j.bmcl.2013.08.074

Entry authors: Giannetti, A.M., Zheng, X., Skelton, N., Wang, W., Bravo, B., Feng, Y., Gunzner-Toste, J., Ho, Y., Hua, R., Wang, C., Zhao, Q., Liederer, B.M., Liu, Y., O'Brien, T., Oeh, J., Sampath, D., Shen, Y., Wang, L., Wu, H., Xiao, Y., Yuen, P., Zak, M., Zhao, G., Dragovich, P.S.

Initial deposition on: 26 July 2013

Initial release on: 25 September 2013

Latest revision on: 28 February 2024

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Structure coordinates (PDB)

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