PDB Entry - 4MR6 (pdb_00004mr6)
(Status - Released)Summary information:
Title: Crystal Structure of the second bromodomain of human BRD2 in complex with a quinazolinone ligand (RVX-208)
PDB DOI: https://doi.org/10.2210/pdb4mr6/pdb
Primary publication DOI: https://doi.org/10.1073/pnas.1310658110
Entry authors: Filippakopoulos, P., Picaud, S., Felletar, I., Martin, S., Fedorov, O., von Delft, F., Arrowsmith, C.H., Edwards, A.M., Weigelt, J., Bountra, C., Knapp, S., Structural Genomics Consortium (SGC)
Initial deposition on: 17 September 2013
Initial release on: 27 November 2013
Latest revision on: 20 September 2023
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Structure coordinates (PDB)
Structure coordinates (PDBML)
X-ray diffraction data (PDBx/mmCIF)
Validation report (mmCIF)
Validation report (XML)
Validation report (PDF)
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