PDB Entry - 4RG0

(Status - Released)

Summary information:

Title: Crystal structure of BTK kinase domain complexed with 2-[8-fluoro-2-[2-(hydroxymethyl)-3-[1-methyl-5-[[5-(4-methylpiperazin-1-yl)-2-pyridyl]amino]-6-oxo-3-pyridyl]phenyl]-1-oxo-3,4-dihydroisoquinolin-6-yl]-2-methyl-propanenitrile

PDB DOI: https://doi.org/10.2210/pdb4rg0/pdb

Primary publication DOI: https://doi.org/10.1016/j.bmcl.2014.11.030

Entry authors: Kuglstatter, A., Wong, A.

Initial deposition on: 29 September 2014

Initial release on: 24 December 2014

Latest revision on: 20 September 2023

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Structure coordinates (PDBx/mmCIF)

Structure coordinates (PDBML)

Structure coordinates (PDB)

X-ray diffraction data (PDBx/mmCIF)

Validation report (mmCIF)

Validation report (PDF)

Validation report (XML)

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