PDB Entry - 4X2I

(Status - Released)

Summary information:

Title: Discovery of benzotriazolo diazepines as orally-active inhibitors of BET bromodomains: Crystal structure of BRD4 with CPI-13

PDB DOI: https://doi.org/10.2210/pdb4x2i/pdb

Primary publication DOI: https://doi.org/10.1021/ml500411h

Entry authors: Bellon, S.F., Jayaram, H., Poy, F.

Initial deposition on: 26 November 2014

Initial release on: 11 November 2015

Latest revision on: 28 February 2024