PDB Entry - 4X7H

(Status - Released)

Summary information:

Title: Co-crystal Structure of PERK bound to N-{5-[(6,7-dimethoxyquinolin-4-yl)oxy]pyridin-2-yl}-1-methyl-3-oxo-2-phenyl-5-(pyridin-4-yl)-2,3-dihydro-1H-pyrazole-4-carboxamide inhibitor

PDB DOI: https://doi.org/10.2210/pdb4x7h/pdb

Primary publication DOI: https://doi.org/10.1021/jm5017494

Entry authors: Shaffer, P.L., Bellon, S.F., Long, A.M., Chen, H.

Initial deposition on: 9 December 2014

Initial release on: 4 February 2015

Latest revision on: 27 September 2023

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Structure coordinates (PDBx/mmCIF)

Structure coordinates (PDBML)

Structure coordinates (PDB)

X-ray diffraction data (PDBx/mmCIF)

Validation report (XML)

Validation report (PDF)

Validation report (mmCIF)

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