PDB Entry - 4X7N

(Status - Released)

Summary information:

Title: Co-crystal Structure of PERK bound to 4-[2-amino-4-methyl-3-(2-methylquinolin-6-yl)benzoyl]-1-methyl-2,5-diphenyl-1,2-dihydro-3H-pyrazol-3-one inhibitor

PDB DOI: https://doi.org/10.2210/pdb4x7n/pdb

Primary publication DOI: https://doi.org/10.1021/jm5017494

Entry authors: Shaffer, P.L., Long, A.M., Chen, H.

Initial deposition on: 9 December 2014

Initial release on: 28 January 2015

Latest revision on: 27 September 2023

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Structure coordinates (PDBx/mmCIF)

Structure coordinates (PDBML)

Structure coordinates (PDB)

X-ray diffraction data (PDBx/mmCIF)

Validation report (XML)

Validation report (mmCIF)

Validation report (PDF)

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