PDB Entry - 5A9U

(Status - Released)

Summary information:

Title: Structure of C1156Y Mutant Human Anaplastic Lymphoma Kinase in Complex with PF-06463922 ((10R)-7-amino-12-fluoro-2,10,16-trimethyl- 15-oxo-10,15,16,17-tetrahydro-2H-8,4-(metheno)pyrazolo(4,3-h)(2,5,11) benzoxadiazacyclotetradecine-3-carbonitrile).

PDB DOI: https://doi.org/10.2210/pdb5a9u/pdb

Primary publication DOI: https://doi.org/10.1056/NEJMOA1508887

Entry authors: McTigue, M., Deng, Y.-L., Liu, W., Brooun, A., Stewart, A.

Initial deposition on: 22 July 2015

Initial release on: 8 June 2016

Latest revision on: 10 January 2024

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Structure coordinates (PDB)

X-ray diffraction data (PDBx/mmCIF)

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Validation report (XML)

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