PDB Entry - 5DT2

(Status - Released)

Summary information:

Title: Crystal structure of Dot1L in complex with inhibitor CPD11 [N4-methyl-N2-(2-methyl-1-(2-phenoxyphenyl)-1H-indol-6-yl)pyrimidine-2,4-diamine]

PDB DOI: https://doi.org/10.2210/pdb5dt2/pdb

Primary publication DOI: https://doi.org/10.1021/acsmedchemlett.6b00167

Entry authors: Scheufler, C., Gaul, C., Be, C., Moebitz, H.

Initial deposition on: 17 September 2015

Initial release on: 15 June 2016

Latest revision on: 10 January 2024

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Structure coordinates (PDBx/mmCIF)

Structure coordinates (PDBML)

Structure coordinates (PDB)

X-ray diffraction data (PDBx/mmCIF)

Validation report (XML)

Validation report (PDF)

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