PDB Entry - 5EI4
(Status - Released)Summary information:
Title: First domain of human bromodomain BRD4 in complex with inhibitor 8-(5-Amino-1H-[1,2,4]triazol-3-ylsulfanylmethyl)-3-(4-chlorobenzyl)-7-ethyl-3,7-dihydropurine-2,6-dione
PDB DOI: https://doi.org/10.2210/pdb5ei4/pdb
Primary publication DOI: https://doi.org/10.1021/acs.jmedchem.5b01708
Entry authors: Raux, B., Rebuffet, E., Betzi, S., Morelli, X.
Initial deposition on: 29 October 2015
Initial release on: 20 January 2016
Latest revision on: 10 January 2024
Downloads:
Structure coordinates (PDBx/mmCIF)
Structure coordinates (PDBML)
Structure coordinates (PDB)
X-ray diffraction data (PDBx/mmCIF)
Validation report (PDF)
Validation report (XML)
Links to more resources for 5EI4 at: