PDB Entry - 5EI4

(Status - Released)

Summary information:

Title: First domain of human bromodomain BRD4 in complex with inhibitor 8-(5-Amino-1H-[1,2,4]triazol-3-ylsulfanylmethyl)-3-(4-chlorobenzyl)-7-ethyl-3,7-dihydropurine-2,6-dione

PDB DOI: https://doi.org/10.2210/pdb5ei4/pdb

Primary publication DOI: https://doi.org/10.1021/acs.jmedchem.5b01708

Entry authors: Raux, B., Rebuffet, E., Betzi, S., Morelli, X.

Initial deposition on: 29 October 2015

Initial release on: 20 January 2016

Latest revision on: 10 January 2024

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Structure coordinates (PDBx/mmCIF)

Structure coordinates (PDBML)

Structure coordinates (PDB)

X-ray diffraction data (PDBx/mmCIF)

Validation report (PDF)

Validation report (XML)

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