PDB Entry - 5EM5

(Status - Released)

Summary information:

Title: EGFR kinase domain mutant ""TMLR"" with pyridone compound 2: 4-[2-(4-chlorophenyl)ethylamino]-~{N}-[4-(4-methylpiperazin-1-yl)phenyl]-2-oxidanylidene-1~{H}-pyridine-3-carboxamide

PDB DOI: https://doi.org/10.2210/pdb5em5/pdb

Primary publication DOI: https://doi.org/10.1021/acsmedchemlett.5b00428

Entry authors: Eigenbrot, C., Yu, C.

Initial deposition on: 5 November 2015

Initial release on: 30 December 2015

Latest revision on: 6 March 2024

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Structure coordinates (PDBx/mmCIF)

Structure coordinates (PDBML)

Structure coordinates (PDB)

X-ray diffraction data (PDBx/mmCIF)

Validation report (PDF)

Validation report (XML)

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