PDB Entry - 5FI4

(Status - Released)

Summary information:

Title: Discovery of imidazo[1,2-a]-pyridine inhibitors of pan-PI3 kinases that are efficacious in a mouse xenograft model

PDB DOI: https://doi.org/10.2210/pdb5fi4/pdb

Primary publication DOI: https://doi.org/10.1016/j.bmcl.2016.01.003

Entry authors: Elling, R.A., Knapp, M.S., Han, W., Daniel, L.M., Xy, Y., Burger, M.T., Ni, Z., Smith, A., Lan, J., Williams, T., Verhagen, J., Huh, K., Merritt, H., Chan, J., Kaufman, S., Voliva, C.F., Pecchi, S.

Initial deposition on: 22 December 2015

Initial release on: 3 February 2016

Latest revision on: 6 March 2024

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Structure coordinates (PDB)

X-ray diffraction data (PDBx/mmCIF)

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