PDB Entry - 5HG9

(Status - Released)

Summary information:

Title: EGFR (L858R, T790M, V948R) in complex with 1-[(3R,4R)-3-[({2-[(1-methyl-1H-pyrazol-4-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-4-yl}oxy)methyl]-4-(trifluoromethyl)pyrrolidin-1-yl]prop-2-en-1-one

PDB DOI: https://doi.org/10.2210/pdb5hg9/pdb

Primary publication DOI: https://doi.org/10.1021/acs.jmedchem.5b01633

Entry authors: Gajiwala, K.S.

Initial deposition on: 8 January 2016

Initial release on: 3 February 2016

Latest revision on: 23 March 2016

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Structure coordinates (PDBx/mmCIF)

Structure coordinates (PDBML)

Structure coordinates (PDB)

X-ray diffraction data (PDBx/mmCIF)

Validation report (PDF)

Validation report (XML)

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