PDB Entry - 5I2R (pdb_00005i2r)

(Status - Released)

Summary information:

Title: CRYSTAL STRUCTURE OF HUMAN PHOSPHODIESTERASE 10 IN COMPLEX WITH C2(=NN(c1cccc(c1)OC(F)(F)F)C=CC2=O)c3ccnn3c4ccccc4, micromolar IC50=0.019462

PDB DOI: https://doi.org/10.2210/pdb5i2r/pdb

Primary publication DOI: https://doi.org/10.1021/acs.jmedchem.5b01875

Entry authors: Joseph, C., Koerner, M., Rudolph, M.G.

Initial deposition on: 9 February 2016

Initial release on: 9 March 2016

Latest revision on: 16 October 2024

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Structure coordinates (PDBx/mmCIF)

Structure coordinates (PDB)

Structure coordinates (PDBML)

X-ray diffraction data (PDBx/mmCIF)

Validation report (XML)

Validation report (mmCIF)

Validation report (PDF)

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