PDB Entry - 5I96

(Status - Released)

Summary information:

Title: Crystal Structure of Human Mitochondrial Isocitrate Dehydrogenase (IDH2) R140Q Mutant Homodimer in Complex with AG-221 (Enasidenib) Inhibitor.

PDB DOI: https://doi.org/10.2210/pdb5i96/pdb

Primary publication DOI: https://doi.org/10.1158/2159-8290.CD-16-1034

Entry authors: Wei, W., Zhang, B., Jin, L., Jiang, F., DeLaBarre, B., Travins, J.A., Padyana, A.K.

Initial deposition on: 19 February 2016

Initial release on: 8 March 2017

Latest revision on: 27 September 2023

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Structure coordinates (PDBx/mmCIF)

Structure coordinates (PDBML)

Structure coordinates (PDB)

X-ray diffraction data (PDBx/mmCIF)

Validation report (mmCIF)

Validation report (XML)

Validation report (PDF)

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