PDB Entry - 5KDH

(Status - Released)

Summary information:

Title: CRYSTAL STRUCTURE OF THE FIRST BROMODOMAIN OF HUMAN BRD4 IN COMPLEX WITH A DIHYDROPYRIDOPYRIMIDINE SCAFFOLD INHIBITOR

PDB DOI: https://doi.org/10.2210/pdb5kdh/pdb

Primary publication DOI: https://doi.org/10.1021/acs.jmedchem.6b01336

Entry authors: Zhu, J.-Y., Schonbrunn, E.

Initial deposition on: 8 June 2016

Initial release on: 2 August 2017

Latest revision on: 27 September 2023

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Structure coordinates (PDB)

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Validation report (mmCIF)

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