PDB Entry - 5KYK

(Status - Released)

Summary information:

Title: Covalent GTP-competitive inhibitors of KRAS G12C: Guanosine bisphosphonate Analogs

PDB DOI: https://doi.org/10.2210/pdb5kyk/pdb

Primary publication DOI: https://doi.org/10.1021/acsmedchemlett.6b00373

Entry authors: Xiong, Y., Lu, J., Hunter, J., Li, L., Scott, D., Manandhar, A., Gondi, S., Westover, K.D., Gray, N.S.

Initial deposition on: 21 July 2016

Initial release on: 12 April 2017

Latest revision on: 4 October 2023

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