PDB Entry - 5LJ2

(Status - Released)

Summary information:

Title: N-TERMINAL BROMODOMAIN OF HUMAN BRD4 WITH 5-(5-aminopyridin-3-yl)-8-(((3R,4R)-3-((1,1-dioxidotetrahydro-2H-thiopyran-4-yl)methoxy)piperidin-4-yl)amino)-3-methyl-1,7-naphthyridin-2(1H)-one

PDB DOI: https://doi.org/10.2210/pdb5lj2/pdb

Primary publication DOI: https://doi.org/10.1002/anie.201603928

Entry authors: Chung, C., Bamborough, P., Demont, E.

Initial deposition on: 17 July 2016

Initial release on: 31 August 2016

Latest revision on: 14 September 2016

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Structure coordinates (PDBx/mmCIF)

Structure coordinates (PDBML)

Structure coordinates (PDB)

X-ray diffraction data (PDBx/mmCIF)

Validation report (PDF)

Validation report (XML)

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