PDB Entry - 5UGA
(Status - Released)Summary information:
Title: Crystal structure of the EGFR kinase domain (L858R, T790M, V948R) in complex with 4-(4-{[2-{[(3S)-1-acetylpyrrolidin-3-yl]amino}-9-(propan-2-yl)-9H-purin-6-yl]amino}phenyl)-1-methylpiperazin-1-ium
PDB DOI: https://doi.org/10.2210/pdb5uga/pdb
Primary publication DOI: https://doi.org/10.1021/acs.jmedchem.6b01894
Entry authors: Gajiwala, K.S., Ferre, R.A.
Initial deposition on: 7 January 2017
Initial release on: 22 March 2017
Latest revision on: 6 March 2024
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Structure coordinates (PDBx/mmCIF)
Structure coordinates (PDBML)
Structure coordinates (PDB)
X-ray diffraction data (PDBx/mmCIF)
Validation report (PDF)
Validation report (XML)
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