PDB Entry - 5UK8

(Status - Released)

Summary information:

Title: The co-structure of (R)-4-(6-(1-(cyclopropylsulfonyl)cyclopropyl)-2-(1H-indol-4-yl)pyrimidin-4-yl)-3-methylmorpholine and a rationally designed PI3K-alpha mutant that mimics ATR

PDB DOI: https://doi.org/10.2210/pdb5uk8/pdb

Primary publication DOI: https://doi.org/10.1016/j.jmb.2017.04.006

Entry authors: Knapp, M.S., Mamo, M., Elling, R.A.

Initial deposition on: 20 January 2017

Initial release on: 14 June 2017

Latest revision on: 3 April 2024

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Structure coordinates (PDBx/mmCIF)

Structure coordinates (PDBML)

Structure coordinates (PDB)

X-ray diffraction data (PDBx/mmCIF)

Validation report (XML)

Validation report (PDF)

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