PDB Entry - 5UKJ

(Status - Released)

Summary information:

Title: The co-structure of N,N-dimethyl-4-[(6R)-6-methyl-5-(1H-pyrrolo[2,3- b]pyridin-4-yl)-4,5,6,7-tetrahydropyrazolo[1,5- a]pyrazin-3-yl]benzenesulfonamide and a rationally designed PI3K-alpha mutant that mimics ATR

PDB DOI: https://doi.org/10.2210/pdb5ukj/pdb

Primary publication DOI: https://doi.org/10.1016/j.jmb.2017.04.006

Entry authors: Knapp, M.S., Elling, R.A., Mamo, M.

Initial deposition on: 23 January 2017

Initial release on: 10 May 2017

Latest revision on: 3 April 2024

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Structure coordinates (PDBx/mmCIF)

Structure coordinates (PDBML)

Structure coordinates (PDB)

X-ray diffraction data (PDBx/mmCIF)

Validation report (XML)

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