PDB Entry - 5UOY

(Status - Released)

Summary information:

Title: Crystal structure of human PDE1B catalytic domain in complex with inhibitor 16j (6-(4-Methoxybenzyl)-9-((tetrahydro-2H-pyran-4-yl)methyl)-8,9,10,11-tetrahydropyrido[4',3':4,5]thieno[3,2-e][1,2,4]triazolo[1,5-c]pyrimidin-5(6H)-one)

PDB DOI: https://doi.org/10.2210/pdb5uoy/pdb

Primary publication DOI: https://doi.org/10.1021/acs.jmedchem.7b00302

Entry authors: Cedervall, E.P., Allerston, C.K., Xu, R., Sridhar, V., Barker, R., Aertgeerts, K.

Initial deposition on: 1 February 2017

Initial release on: 26 April 2017

Latest revision on: 4 October 2023

Downloads:

Structure coordinates (PDBx/mmCIF)

Structure coordinates (PDBML)

Structure coordinates (PDB)

X-ray diffraction data (PDBx/mmCIF)

Validation report (mmCIF)

Validation report (PDF)

Validation report (XML)

Links to more resources for 5UOY at: