PDB Entry - 5V7I

(Status - Released)

Summary information:

Title: Crystal structure of homo sapiens serine hydroxymethyltransferase 2 (mitochondrial) (SHMT2), in complex with glycine, PLP and folate-competitive pyrazolopyran inhibitor: 6-amino-4-isopropyl-3-methyl-4-(3-(pyrrolidin-1-yl)-5-(trifluoromethyl)phenyl)-1,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile

PDB DOI: https://doi.org/10.2210/pdb5v7i/pdb

Primary publication DOI: https://doi.org/10.1073/pnas.1706617114

Entry authors: Ducker, G.S., Ghergurovich, J.M., Mainolfi, N., Suri, V., Jeong, S., Friedman, A., Manfredi, M., Kim, H., Rabinowitz, J.D.

Initial deposition on: 20 March 2017

Initial release on: 11 October 2017

Latest revision on: 15 November 2023

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Structure coordinates (PDBx/mmCIF)

Structure coordinates (PDBML)

Structure coordinates (PDB)

X-ray diffraction data (PDBx/mmCIF)

Validation report (XML)

Validation report (PDF)

Validation report (mmCIF)

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