PDB Entry - 5V9P

(Status - Released)

Summary information:

Title: Crystal structure of pyrrolidine amide inhibitor [(3S)-3-(4-bromo-1H-pyrazol-1-yl)pyrrolidin-1-yl][3-(propan-2-yl)-1H-pyrazol-5-yl]methanone (compound 35) in complex with KDM5A

PDB DOI: https://doi.org/10.2210/pdb5v9p/pdb

Primary publication DOI: https://doi.org/10.1016/j.bmcl.2017.05.016

Entry authors: Kiefer, J.R., Liang, J., Vinogradova, M.

Initial deposition on: 23 March 2017

Initial release on: 10 May 2017

Latest revision on: 4 October 2023

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Structure coordinates (PDBx/mmCIF)

Structure coordinates (PDBML)

Structure coordinates (PDB)

X-ray diffraction data (PDBx/mmCIF)

Validation report (XML)

Validation report (PDF)

Validation report (mmCIF)

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