PDB Entry - 6FT3

(Status - Released)

Summary information:

Title: Crystal Structure of the first bromodomain of human BRD4 in complex with a 3,5-dimethylisoxazol ligand

PDB DOI: https://doi.org/10.2210/pdb6ft3/pdb

Primary publication DOI: https://doi.org/10.1016/j.bmc.2018.05.003

Entry authors: Filippakopoulos, P., Picaud, S., Pike, A.C.W., Krojer, T., Conway, S.J., von Delft, F., Arrowsmith, C.H., Edwards, A.M., Bountra, C., Structural Genomics Consortium (SGC)

Initial deposition on: 20 February 2018

Initial release on: 18 April 2018

Latest revision on: 17 January 2024

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Structure coordinates (PDBx/mmCIF)

Structure coordinates (PDBML)

Structure coordinates (PDB)

X-ray diffraction data (PDBx/mmCIF)

Validation report (PDF)

Validation report (XML)

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