PDB Entry - 6IAR

(Status - Released)

Summary information:

Title: Tricyclic indazoles a novel class of selective estrogen receptor degrader antagonists

PDB DOI: https://doi.org/10.2210/pdb6iar/pdb

Primary publication DOI: https://doi.org/10.1021/acs.jmedchem.8b01837

Entry authors: Scott, J.S., Bailey, A., Buttar, D., Carbajo, R.J., Curwen, J., Davies, R.D.M., Degorce, S.L., Donald, C., Gangl, E., Greenwood, R., Groombridge, S.D., Johnson, T., Lamont, S., Lawson, M., Lister, A., Morrow, C., Moss, T., Pink, J.H., Polanski, R.

Initial deposition on: 27 November 2018

Initial release on: 23 January 2019

Latest revision on: 24 April 2019

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Structure coordinates (PDB)

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