PDB Entry - 6TPE
(Status - Released)Summary information:
Title: Fragment-based discovery of pyrazolopyridones as JAK1 inhibitors with excellent subtype selectivity
PDB DOI: https://doi.org/10.2210/pdb6tpe/pdb
Primary publication DOI: https://doi.org/10.1021/acs.jmedchem.0c00359
Entry authors: Hansen, B.B., Jepsen, T.H., Larsen, M., Sindet, R., Vifian, T., Burhardt, M.N., Larsen, J., Seitzberg, J.G., Carnerup, M.A., Jerre, A., Molck, C., Rai, S., Nasipireddy, V.R., Jestel, A., Lammens, A., Ritzen, A.
Initial deposition on: 13 December 2019
Initial release on: 10 June 2020
Latest revision on: 22 July 2020
Downloads:
Structure coordinates (PDBx/mmCIF)
Structure coordinates (PDBML)
Structure coordinates (PDB)
X-ray diffraction data (PDBx/mmCIF)
Validation report (PDF)
Validation report (XML)
Links to more resources for 6TPE at: