PDB Entry - 6TPE

(Status - Released)

Summary information:

Title: Fragment-based discovery of pyrazolopyridones as JAK1 inhibitors with excellent subtype selectivity

PDB DOI: https://doi.org/10.2210/pdb6tpe/pdb

Primary publication DOI: https://doi.org/10.1021/acs.jmedchem.0c00359

Entry authors: Hansen, B.B., Jepsen, T.H., Larsen, M., Sindet, R., Vifian, T., Burhardt, M.N., Larsen, J., Seitzberg, J.G., Carnerup, M.A., Jerre, A., Molck, C., Rai, S., Nasipireddy, V.R., Jestel, A., Lammens, A., Ritzen, A.

Initial deposition on: 13 December 2019

Initial release on: 10 June 2020

Latest revision on: 22 July 2020

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Structure coordinates (PDBx/mmCIF)

Structure coordinates (PDBML)

Structure coordinates (PDB)

X-ray diffraction data (PDBx/mmCIF)

Validation report (PDF)

Validation report (XML)

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