PDB Entry - 7G3S (pdb_00007g3s)
(Status - Released)Summary information:
Title: Crystal Structure of rat Autotaxin in complex with 2-[(5-chloro-2,3-dihydro-1H-inden-2-yl)amino]-6-(oxetan-3-yl)-7H-pyrrolo[3,4-d]pyrimidin-5-one, i.e. SMILES O=C1N(C2COC2)Cc2nc(N[C@H]3Cc4c(C3)ccc(c4)Cl)ncc12 with IC50=0.150181 microM
PDB DOI: https://doi.org/10.2210/pdb7g3s/pdb
Entry authors: Stihle, M., Benz, J., Hunziker, D., Pinard, E., Rudolph, M.G.
Initial deposition on: 5 June 2023
Initial release on: 18 December 2024
Latest revision on: 18 December 2024
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Structure coordinates (PDBx/mmCIF)
Structure coordinates (PDB)
Structure coordinates (PDBML)
X-ray diffraction data (PDBx/mmCIF)
Validation report (mmCIF)
Validation report (PDF)
Validation report (XML)
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