PDB Entry - 7KHH

(Status - Released)

Summary information:

Title: Ternary complex of VHL/BRD4-BD1/Compound9 (4-(3,5-difluoropyridin-2-yl)-N-(11-(((S)-1-((2S,4R)-4-hydroxy-2-((4-(4-methylthiazol-5-yl)benzyl)carbamoyl)pyrrolidin-1-yl)-3,3-dimethyl-1-oxobutan-2-yl)amino)-11-oxoundecyl)-10-methyl-7-((methylsulfonyl)methyl)-11-oxo-3,4,10,11-tetrahydro-1H-1,4,10-triazadibenzo[cd,f]azulene-6-carboxamide)

PDB DOI: https://doi.org/10.2210/pdb7khh/pdb

Primary publication DOI: https://doi.org/10.1021/acs.jmedchem.0c01846

Entry authors: Murray, J.M.

Initial deposition on: 21 October 2020

Initial release on: 24 February 2021

Latest revision on: 18 October 2023

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Structure coordinates (PDBx/mmCIF)

Structure coordinates (PDBML)

Structure coordinates (PDB)

X-ray diffraction data (PDBx/mmCIF)

Validation report (XML)

Validation report (mmCIF)

Validation report (PDF)

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