PDB Entry - 7MCF

(Status - Released)

Summary information:

Title: CRYSTAL STRUCTURE OF THE FIRST BROMODOMAIN OF HUMAN BRD4 IN COMPLEX WITH 2-{3-(1,4-dimethyl-1H-1,2,3-triazol-5-yl)-6-fluoro-5-[(S)-(3-fluoropyridin-2-yl)(oxan-4-yl)methyl]-5H-pyrido[3,2-b]indol-7-yl}propan-2-ol

PDB DOI: https://doi.org/10.2210/pdb7mcf/pdb

Primary publication DOI: https://doi.org/10.1016/j.bmcl.2021.128108

Entry authors: Sheriff, S.

Initial deposition on: 2 April 2021

Initial release on: 26 May 2021

Latest revision on: 18 October 2023

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Structure coordinates (PDBx/mmCIF)

Structure coordinates (PDBML)

Structure coordinates (PDB)

X-ray diffraction data (PDBx/mmCIF)

Validation report (PDF)

Validation report (XML)

Validation report (mmCIF)

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