PDB Entry - 7UZN

(Status - Released)

Summary information:

Title: CRYSTAL STRUCTURE OF THE FIRST BROMODOMAIN OF HUMAN BRD4 IN COMPLEX WITH BMT-206059 AKA 2-{(3M)-3-(1,4-DIMETHYL-1H-1,2,3-TRIAZOL-5-YL)-8-FLUORO-5-[(S)-(OXAN-4-YL)(PHENYL)METHYL]-5H-PYRIDO[3,2-b]INDOL-7-YL}PROPAN-2-OL, TRIPLY DEUTERATED ON THE 4-METHYL GROUP

PDB DOI: https://doi.org/10.2210/pdb7uzn/pdb

Primary publication DOI: https://doi.org/10.1021/acsmedchemlett.2c00219

Entry authors: Sheriff, S.

Initial deposition on: 9 May 2022

Initial release on: 17 August 2022

Latest revision on: 18 October 2023

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Structure coordinates (PDBx/mmCIF)

Structure coordinates (PDBML)

Structure coordinates (PDB)

X-ray diffraction data (PDBx/mmCIF)

Validation report (XML)

Validation report (mmCIF)

Validation report (PDF)

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