PDB Entry - 8EAD

(Status - Released)

Summary information:

Title: Crystal structure of the first bromodomain (BD1) of human BRD4 in complex with dual BRD4-JAK2 inhibitor MA9-177

PDB DOI: https://doi.org/10.2210/pdb8ead/pdb

Entry authors: Karim, M.R., Schonbrunn, E.

Initial deposition on: 29 August 2022

Initial release on: 7 September 2022

Latest revision on: 18 October 2023

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Structure coordinates (PDBx/mmCIF)

Structure coordinates (PDBML)

Structure coordinates (PDB)

X-ray diffraction data (PDBx/mmCIF)

Validation report (mmCIF)

Validation report (XML)

Validation report (PDF)

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