PDB Entry - 8FJZ

(Status - Released)

Summary information:

Title: Crystal structure of HPK1 kinase domain T165E,S171E phosphomimetic mutant in complex with 3-{4-[(3R,5S)-3-Amino-5-methylpiperidin-1-yl]-6-chloro-7H-pyrrolo[2,3-d]pyrimidin-5-yl}benzonitrile

PDB DOI: https://doi.org/10.2210/pdb8fjz/pdb

Primary publication DOI: https://doi.org/10.1021/acs.jmedchem.2c02038

Entry authors: McTigue, M., Johnson, E., Cronin, C.

Initial deposition on: 20 December 2022

Initial release on: 5 April 2023

Latest revision on: 25 October 2023

Downloads:

Structure coordinates (PDBx/mmCIF)

Structure coordinates (PDBML)

Structure coordinates (PDB)

X-ray diffraction data (PDBx/mmCIF)

Validation report (mmCIF)

Validation report (XML)

Validation report (PDF)

Links to more resources for 8FJZ at: