PDB Entry - 8G3E (pdb_00008g3e)

(Status - Released)

Summary information:

Title: Crystal structure of human WDR5 in complex with (1M)-N-[(3,5-difluoro[1,1'-biphenyl]-4-yl)methyl]-6-methyl-4-oxo-1-(pyridin-3-yl)-1,4-dihydropyridazine-3-carboxamide (compound 2, WDR5-MYC inhibitor)

PDB DOI: https://doi.org/10.2210/pdb8g3e/pdb

Primary publication DOI: https://doi.org/10.1021/acs.jmedchem.3c00787

Entry authors: Zhao, M.

Initial deposition on: 7 February 2023

Initial release on: 28 June 2023

Latest revision on: 25 October 2023

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Structure coordinates (PDBx/mmCIF)

Structure coordinates (PDB)

Structure coordinates (PDBML)

X-ray diffraction data (PDBx/mmCIF)

Validation report (mmCIF)

Validation report (PDF)

Validation report (XML)

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