PDB Entry - 8HLR (pdb_00008hlr)

(Status - Released)

Summary information:

Title: Human ADP-ribosyltransferase 1 (PARP1) catalytic domain bound to Fluzoparib (SHR3162)

PDB DOI: https://doi.org/10.2210/pdb8hlr/pdb

Primary publication DOI: https://doi.org/10.1016/j.bioorg.2025.108471

Entry authors: Wang, X.Y., Zhou, J., Xu, B.L.

Initial deposition on: 30 November 2022

Initial release on: 1 May 2024

Latest revision on: 14 May 2025

Downloads:

Structure coordinates (PDBx/mmCIF)

Structure coordinates (PDB)

Structure coordinates (PDBML)

X-ray diffraction data (PDBx/mmCIF)

Validation report (PDF)

Validation report (XML)

Validation report (mmCIF)

Links to more resources for 8HLR (pdb_00008hlr) at: